Product Overview
5-BDBD | T22518 | TargetMol Chemicals
CAS: 768404-03-1
Smiles: Brc1cccc(c1)C1=NCC(=O)Nc2c1oc1ccccc21
Formula: C17H11BrN2O2
Pathway: Membrane transporter/Ion channel|||Neuroscience
Target: P2X Receptor|||P2 Receptor
Receptor: N/A
Bioactivity: 5-BDBD is a potent and selective P2X4 receptor antagonist. 5-BDBD inhibits rP2X4R-mediated currents with an IC50 of 0.75 μM. 5-BDBD completely blocked the basal and acute hyperalgesia induced by NTG.
Molecular Weight: 355, 191
