Product Overview
APY0201 | T2061 | TargetMol Chemicals
CAS: 1232221-74-7
Smiles: Cc1cccc(\C=N\Nc2cc(N3CCOCC3)n3nc(cc3n2)-c2ccncc2)c1
Formula: C23H23N7O
Pathway: Immunology/Inflammation|||PI3K/Akt/mTOR signaling
Target: PI3K|||Interleukin
Receptor: N/A
Bioactivity: APY0201 is a effective, highly specific, ATP-competitive PIKfyve inhibitor (IC50: 5.2 nM). It can interrupt the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns(3, 5)P2.
Molecular Weight: 413, 485
