Product Overview
AZD1981 | T6399 | TargetMol Chemicals
CAS: 802904-66-1
Smiles: CC(=O)Nc1cccc2n(CC(O)=O)c(C)c(Sc3ccc(Cl)cc3)c12
Formula: C19H17ClN2O3S
Pathway: Endocrinology/Hormones|||GPCR/G Protein|||Immunology/Inflammation
Target: GPR|||Prostaglandin Receptor
Receptor: N/A
Bioactivity: AZD1981 is an effective and specific CRTh2 (DP2) receptor antagonist (IC50: 4 nM), showing >1000-fold selectivity over more than 340 other enzymes and receptors, including DP1. AZD1981 has been used in trials studying the treatment and basic science of Asthma, Postmenopausal, Pharmakokinetic, Asthma Patients, and Drug Interaction, among others.
Molecular Weight: 388, 87
