Product Overview
BAY1082439 | T14511 | TargetMol Chemicals
CAS: 1375469-38-7
Smiles: COc1c(OC[C@H](O)CN2CCOCC2)ccc2C3=NCCN3C(NC(=O)c3cccnc3C)=Nc12
Formula: C25H30N6O5
Pathway: Apoptosis|||PI3K/Akt/mTOR signaling
Target: Apoptosis|||PI3K
Receptor: N/A
Bioactivity: BAY1082439 is highly effective in inhibiting Pten-null prostate cancer growth[1][2] and it is an orally bioavailable, selective PI3Kα/β/δ inhibitor. BAY1082439 also inhibits mutated forms of PIK3CA.
Molecular Weight: 494, 552