Product Overview
BD 1008 dihydrobromide | T21788 | TargetMol Chemicals
CAS: 138356-09-9
Smiles: Br.Br.CN(CCN1CCCC1)CCc1ccc(Cl)c(Cl)c1
Formula: N/A
Pathway: GPCR/G Protein
Target: Sigma receptor
Receptor: N/A
Bioactivity: BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. BD1008 dihydrobromide attenuate the toxicity and stimulant effects of cocaine through antagonism of sigma receptors[1].
Molecular Weight: 463, 078