Product Overview
BETd-260 | T14550 | TargetMol Chemicals
CAS: 2093388-62-4
Smiles: CCn1nc(cc1Nc1nc(nc2[nH]c3cc(-c4c(C)noc4C)c(OC)cc3c12)C(=O)NCCCCCc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O)C1CC1
Formula: C43H46N10O6
Pathway: Chromatin/Epigenetic|||Others
Target: Others|||Epigenetic Reader Domain
Receptor: N/A
Bioactivity: BETd-260 is a potent degrader of BET based on PROTAC technology, with as low as 30 pM against BRD4 protein in RS4;11 leukemia cell line.
Molecular Weight: 798, 905
