Product Overview
Bitopertin | T6788 | TargetMol Chemicals
CAS: 845614-11-1
Smiles: C[C@H](Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
Formula: C21H20F7N3O4S
Pathway: Neuroscience
Target: GlyT
Receptor: N/A
Bioactivity: Bitopertin (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nM in Chinese hamster ovary cells.
Molecular Weight: 543, 46