Product Overview
BMS-819881 | T14678 | TargetMol Chemicals
CAS: 1197420-05-5
Smiles: COc1cc(ccc1OC[C@H](O)C1CC1)-n1cnc2cc(sc2c1=O)-c1ccc(Cl)cc1
Formula: C24H21ClN2O4S
Pathway: Metabolism
Target: P450
Receptor: N/A
Bioactivity: BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
Molecular Weight: 468, 95
