Product Overview
BMS-986122 | T26869 | TargetMol Chemicals
CAS: 313669-88-4
Smiles: COc1ccc(cc1Br)C1SCCN1S(=O)(=O)c1ccc(Cl)cc1
Formula: C16H15BrClNO3S2
Pathway: Endocrinology/Hormones|||GPCR/G Protein|||Neuroscience
Target: Opioid Receptor
Receptor: N/A
Bioactivity: BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM).
Molecular Weight: 448, 77
