Product Overview
BMS986260 | T8730 | TargetMol Chemicals
CAS: 2001559-19-7
Smiles: OCCn1cnc(c1-c1ccc2ncc(C#N)n2n1)-c1ccc(F)c(Cl)c1
Formula: C18H12ClFN6O
Pathway: Stem Cells
Target: TGF-beta/Smad
Receptor: N/A
Bioactivity: BMS-986260 is a selective, and orally bioavailable TGFβR1 inhibitor(IC50 = 1.6 nM).
Molecular Weight: 382, 78