Product Overview
BPTU | T4132 | TargetMol Chemicals
CAS: 870544-59-5
Smiles: CC(C)(C)c1ccccc1Oc1ncccc1NC(=O)Nc1ccc(OC(F)(F)F)cc1
Formula: C23H22F3N3O3
Pathway: Neuroscience
Target: P2 Receptor
Receptor: N/A
Bioactivity: Allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM). Non-nucleotide ligand. Binds receptor outside of the helical bundle. Blocks inhibition of spontaneous contraction of rat and mouse colon induced by electrical field stimulation, nicotine and P2Y agonists. Antithrombotic; reduces platelet aggregation.
Molecular Weight: 445, 442