Product Overview
BRD7-IN-1 | T17697 | TargetMol Chemicals
CAS: T17697
Smiles: CN1C=C(C2=CC(OC)=C(CN3CCNCC3)C(OC)=C2)C(C=CN=C4)=C4C1=O.Cl.Cl
Formula: C22H28Cl2N4O3
Pathway: Chromatin/Epigenetic|||Others
Target: Others|||Epigenetic Reader Domain
Receptor: N/A
Bioactivity: BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), binds to a VHL ligand via a linker to form a PROTAC VZ185 (VZ185 against BRD7/9 with DC50s of 4.5 and 1.8 nM, respectively).
Molecular Weight: 467, 39
