Product Overview
BX-912 | T1837 | TargetMol Chemicals
CAS: 702674-56-4
Smiles: Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1c[nH]cn1
Formula: C20H23BrN8O
Pathway: Angiogenesis|||Apoptosis|||Cell Cycle/Checkpoint|||PI3K/Akt/mTOR signaling|||Tyrosine Kinase/Adaptors
Target: Apoptosis|||VEGFR|||PKA|||Chk|||CDK|||PDK
Receptor: N/A
Bioactivity: BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM). The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.
Molecular Weight: 471, 363
