Product Overview
CCG-63808 | T14898 | TargetMol Chemicals
CAS: 620113-73-7
Smiles: Cc1cccn2c1nc(Oc1ccc(F)cc1)c(\C=C(/C#N)c1nc3ccccc3s1)c2=O
Formula: C25H15FN4O2S
Pathway: GPCR/G Protein
Target: GTPase
Receptor: N/A
Bioactivity: CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM.
Molecular Weight: 454, 48
