Product Overview
CCG215022 | T3498 | TargetMol Chemicals
CAS: 1813527-81-9
Smiles: CC1=C(C(NC(=O)N1)c1ccc(F)c(c1)C(=O)NCc1ccccn1)C(=O)Nc1ccc2[nH]ncc2c1
Formula: C26H22FN7O3
Pathway: GPCR/G Protein|||Tyrosine Kinase/Adaptors
Target: GRK|||PKA
Receptor: N/A
Bioactivity: CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.
Molecular Weight: 499, 506