Product Overview
CCG258208 | T13714 | TargetMol Chemicals
CAS: 2055990-90-2
Smiles: Fc1ccc(cc1C(=O)NCc1cc[nH]n1)[C@@H]1CCNC[C@H]1COc1ccc2OCOc2c1
Formula: C24H25FN4O4
Pathway: GPCR/G Protein
Target: GRK
Receptor: N/A
Bioactivity: GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
Molecular Weight: 452, 486
