CD161 | T14910

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TMC-T14910
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Product Overview

CD161 | T14910 | TargetMol Chemicals

CAS: 1627716-22-6

Smiles: COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(-c3ccnc4ccccc34)c21

Formula: C26H21N5O2

Pathway: Others

Target: Others

Receptor: N/A

Bioactivity: CD161 is a potent, selective, and orally bioavailable BET bromodomain inhibitor (IC50s: 28.2 nM and 7.2 nM for BRD4 BD1 and BRD4 BD2) with good anticancer activity.

Molecular Weight: 435, 487

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