Product Overview
CDK4-IN-1 | T2082 | TargetMol Chemicals
CAS: 1256963-02-6
Smiles: CC(C)c1[nH]nc(Cl)c1-c1ccnc(Nc2ccc(cn2)N2CCC(CC2)N(C)C)n1
Formula: C22H29ClN8
Pathway: Cell Cycle/Checkpoint
Target: CDK
Receptor: N/A
Bioactivity: CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50=5.265 uM) respectively.
Molecular Weight: 440, 98