Product Overview
CL 218872 | T8572 | TargetMol Chemicals
CAS: 66548-69-4
Smiles: Cc1nnc2ccc(nn12)-c1cccc(c1)C(F)(F)F
Formula: C13H9F3N4
Pathway: Membrane transporter/Ion channel|||Neuroscience
Target: GABA Receptor
Receptor: N/A
Bioactivity: CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for α1, α2, α3, α4, α5 and α6-subunit containing receptors respectively). Orally active anxiolytic and anticonvulsant in vivo.
Molecular Weight: 278, 238
