Product Overview
CMP8 | T14987 | TargetMol Chemicals
CAS: 851107-28-3
Smiles: Oc1ccc2C3=C(C(=O)CCC3(Cc3ccc(Cl)cc3)Cc2c1)c1ccc(OCCN2CCCCC2)cc1
Formula: C33H34ClNO3
Pathway: Endocrinology/Hormones
Target: Estrogen Receptor/ERR|||Estrogen/progestogen Receptor
Receptor: N/A
Bioactivity: CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM, 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, respectively.
Molecular Weight: 528, 09