Product Overview
Conantokin G | TP2060 | TargetMol Chemicals
CAS: 93438-65-4
Smiles:
Formula: C88H138N26O44
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: GluN2B (formally NR2B) selective, competitive antagonist of the NMDA receptor. Blocks NMDA-evoked current in mouse cortical neurons (IC50 = 480 nM); also inhibits NMDA-evoked responses in oocytes expressing GluN2B (formally NR2B), but not GluN2A (formally NR2A), subunits (IC50 ~300 nM). Exhibits neuroprotective properties in vivo and in vitro.
Molecular Weight: 2264, 21
