Product Overview
CP-10 | T13627 | TargetMol Chemicals
CAS: 2366268-80-4
Smiles: CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCN(Cc4cn(CCOCCNc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)CC3)nc2n(C2CCCC2)c1=O
Formula: C44H49N13O7
Pathway: Cell Cycle/Checkpoint
Target: CDK
Receptor: N/A
Bioactivity: CP-10 is a PROTAC with highly selective and remarkable CDK6 degradation (DC50: 2.1 nM). It inhibits the proliferation of several hematopoietic cancer cells including multiple myeloma and can degrade mutated and overexpressed CDK6.
Molecular Weight: 871, 96
