Product Overview
CPYPP | T8527 | TargetMol Chemicals
CAS: 310460-39-0
Smiles: Clc1ccccc1C=CC=C1C(=O)NN(C1=O)c1ccccc1
Formula: C18H13ClN2O2
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: CPYPP is an inhibitor of DOCK2-Rac1 interaction. CPYPP binds to DOCK2 DHR-2 domain and inhibits the guanine nucleotide exchange factor (GEF) activity of DOCK2DHR-2 for Rac1 in a dose-dependent manner(IC50 : 22.8 μM). CPYPP also inhibits DOCK180, DOCK5 and less DOCK9
Molecular Weight: 324, 76