Product Overview
CYM2503 | T8963 | TargetMol Chemicals
CAS: 1308833-36-4
Smiles: Cc1cc(=O)[nH]c2cc(NC(=O)[C@H](CCCCNC(=O)OC(C)(C)C)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc34)ccc12
Formula: C45H55N5O7
Pathway: GPCR/G Protein|||Neuroscience
Target: Neuropeptide Y Receptor
Receptor: N/A
Bioactivity: CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by its inability to displace iodinated galanin, or to induce IP1 accumulation on its own).
Molecular Weight: 777, 963