[D-Arg1, D-Phe5, D-Trp7, 9, Leu11]-Substance P | TP1931

[D-Arg1, D-Phe5, D-Trp7, 9, Leu11]-Substance P | TP1931 | TargetMol Chemicals

CAS: 96736-12-8

Smiles:

Formula: C79H109N19O12

Pathway: N/A

Target: N/A

Receptor: N/A

Bioactivity: Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.

Molecular Weight: 1516, 85