(d(CH2)51, Tyr(Me)2, Arg8)-Vasopressin | TP2136

(d(CH2)51, Tyr(Me)2, Arg8)-Vasopressin | TP2136 | TargetMol Chemicals

CAS: 73168-24-8

Smiles:

Formula: C52H74N14O12S2

Pathway: N/A

Target: N/A

Receptor: N/A

Bioactivity: Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.

Molecular Weight: 1151, 38