d[Cha4]-AVP acetate(500170-27-4 free base) | TP2082L

d[Cha4]-AVP acetate(500170-27-4 free base) | TP2082L | TargetMol Chemicals

CAS: TP2082L

Smiles: O=C(N[C@@H](CC(N)=O)C(N[C@H](C(N1CCC[C@H]1C(N[C@H](C(NCC(N)=O)=O)CCC/N=C(N)\N)=O)=O)CSSCCC(N[C@@H](CC2=CC=C(O)C=C2)C(N[C@@H](CC3=CC=CC=C3)C(N4)=O)=O)=O)=O)[C@@H]4CC5CCCCC5.CC(O)=O

Formula: C52H75N13O13S2

Pathway: GPCR/G Protein

Target: Vasopressin Receptor

Receptor: N/A

Bioactivity: d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.

Molecular Weight: 1154, 37