Product Overview
Darapladib | T6109 | TargetMol Chemicals
CAS: 356057-34-6
Smiles: CCN(CC)CCN(Cc1ccc(cc1)-c1ccc(cc1)C(F)(F)F)C(=O)Cn1c2CCCc2c(=O)nc1SCc1ccc(F)cc1
Formula: C36H38F4N4O2S
Pathway: Metabolism
Target: Phospholipase
Receptor: N/A
Bioactivity: Darapladib(IC50=0.25 nM) is a substituted pyrimidone with inhibitory activity towards lipoprotein-associated phospholipase-A2 (Lp-PLA2).
Molecular Weight: 666, 78