Product Overview
DG-041 | T15108 | TargetMol Chemicals
CAS: 861238-35-9
Smiles: Cc1cn(Cc2ccc(Cl)cc2Cl)c2c(\C=C\C(=O)NS(=O)(=O)c3cc(Cl)c(Cl)s3)cc(F)cc12
Formula: C23H15Cl4FN2O3S2
Pathway: GPCR/G Protein|||Immunology/Inflammation|||Others
Target: Others|||Prostaglandin Receptor
Receptor: N/A
Bioactivity: DG-041 is an antagonist of high affinity EP3 receptor (IC50s: 4.6 nM and 8.1 nM in the binding and FLIPR assay, respectively ). DG-041 inhibits PGE2 facilitation of platelet aggregation and it also crosses the blood-brain barrier.
Molecular Weight: 592, 3
