E-4177 | T27229

(No reviews yet) Write a Review
€100.00
SKU:
TMC-T27229
Availability:
IN STOCK
Adding to cart… The item has been added

Product Overview

E-4177 | T27229 | TargetMol Chemicals

CAS: 135070-05-2

Smiles: Cc1ccnc2n(Cc3ccc(cc3)-c3ccccc3C(O)=O)c(nc12)C1CC1

Formula: C24H21N3O2

Pathway: N/A

Target: N/A

Receptor: N/A

Bioactivity: E-4177 is an angiotensin type 1 receptor antagonist. In rat adrenal cortex and liver, E4177 competitively inhibited the specific binding of 125I-[Sar1, Ile8]Ang II, with IC50 being (5.2 +/- 1.0) x 10(-8) M for the adrenal cortex and (1.2 +/- 0.3) x 10(-7) M for the liver.

Molecular Weight: 383, 451

Reviews

(No reviews yet) Write a Review