Product Overview
(E/Z)-IT-603 | T8799 | TargetMol Chemicals
CAS: 292168-90-2
Smiles: COc1cc(Br)cc(\C=C2\NC(=S)NC2=O)c1O
Formula: C11H9BrN2O3S
Pathway: NF-Κb|||Others
Target: Others|||NF-κB
Receptor: N/A
Bioactivity: IT-603 is a cell-permeable c-Rel inhibitor (IC50: 3μM). IT-603 directly and reversibly binds to c-Rel to change its conformation and blocks its DNA binding and transcriptional activity.
Molecular Weight: 329, 17
