Product Overview
ELA-21 (human) | TP2096 | TargetMol Chemicals
CAS: 2245073-05-4
Smiles:
Formula: C112H184N40O25S3
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: High affinity apelin receptor agonist. Binds apelin receptors in left ventricle from normal and pulmonary arterial hypertensive (PAH) hearts (pKi values are 9.31 and 9.46, respectively). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro.
Molecular Weight: 2587, 12
