Product Overview
ELN-441958 | T2086 | TargetMol Chemicals
CAS: 913064-47-8
Smiles: Clc1cccc2CN(C(=O)c12)c1cccc(c1)C(=O)N1CCC2(CC1)CCN(CC2)c1ccncc1
Formula: C29H29ClN4O2
Pathway: GPCR/G Protein
Target: Bradykinin Receptor
Receptor: N/A
Bioactivity: ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958 is highly selective for B1 over B2 receptors.
Molecular Weight: 501, 03
