Product Overview
EN4 | T9061 | TargetMol Chemicals
CAS: 1197824-15-9
Smiles: CCOC1=CC=C(C=C1)OC2=CC=CC=C2NC(=O)C3=CC=C(C=C3)CNC(=O)C=C
Formula: C25H24N2O4
Pathway: Cell Cycle/Checkpoint
Target: c-Myc
Receptor: N/A
Bioactivity: EN4 MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.
Molecular Weight: 416, 47
