Product Overview
EN460 | T15218 | TargetMol Chemicals
CAS: 496807-64-8
Smiles: OC(=O)c1cc(ccc1Cl)N1N=C(\C(=C\c2ccc(o2)-c2ccccc2)C1=O)C(F)(F)F
Formula: C22H12ClF3N2O4
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: EN460 is an inhibitor of endoplasmic reticulum oxidation 1 (ERO1) and interacts selectively (IC50: 1.9 uM) with the reduced, active form of ERO1α and prevents its reoxidation.
Molecular Weight: 460, 79