Product Overview
EPZ004777 | T3081 | TargetMol Chemicals
CAS: 1338466-77-5
Smiles: CC(C)N(CCCNC(=O)Nc1ccc(cc1)C(C)(C)C)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1ccc2c(N)ncnc12
Formula: C28H41N7O4
Pathway: Apoptosis|||Chromatin/Epigenetic
Target: Apoptosis|||Histone Methyltransferase
Receptor: N/A
Bioactivity: EPZ004777 is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.
Molecular Weight: 539, 681
