Product Overview
ERK5-IN-1 | T5184 | TargetMol Chemicals
CAS: 1234479-76-5
Smiles: COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
Formula: C25H29N7O2
Pathway: MAPK
Target: ERK
Receptor: N/A
Bioactivity: ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM). It also inhibits LRRK2[G2019S] (IC50: 26 nM).
Molecular Weight: 459, 554