Product Overview
ERK5-IN-2 | T5535 | TargetMol Chemicals
CAS: 1888305-96-1
Smiles: Fc1cccc(Br)c1C(=O)c1c[nH]c(c1)C(=O)Nc1cccnc1
Formula: C17H11BrFN3O2
Pathway: MAPK
Target: ERK
Receptor: N/A
Bioactivity: ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0.82 μM, 3 μM for ERK5 and ERK5 MEF2D, respectively.
Molecular Weight: 388, 196