Product Overview
Ertiprotafib | T15243 | TargetMol Chemicals
CAS: 251303-04-5
Smiles: Cc1sc2c(Br)c3ccccc3c(-c3cc(C)c(O[C@H](Cc4ccccc4)C(O)=O)c(C)c3)c2c1C
Formula: C31H27BrO3S
Pathway: DNA Damage/DNA Repair|||Metabolism
Target: Phosphatase|||PPAR
Receptor: N/A
Bioactivity: Ertiprotafib is a PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist inhibitor ( IC50s: 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ).
Molecular Weight: 559, 52