Product Overview
Etacstil | T27289 | TargetMol Chemicals
CAS: 155701-61-4
Smiles: CC\C(=C(\c1ccccc1)c1ccc(\C=C\C(O)=O)cc1)c1ccccc1
Formula: C25H22O2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: GW5638 is a estrogen receptor ligand. GW5638 is a prodrug of its active metabolite GW7604. GW5638 appears to act as an antagonist in these in vitro systems, although in a manner distinct from other known ER modulators. GW5638 is also classified as a pseudo-SERD, which could form the basis of a new paradigm of breast cancer hormonal therapy in its own right.
Molecular Weight: 354, 449