Product Overview
GaTx2 | TP2027 | TargetMol Chemicals
CAS: 194665-85-5
Smiles:
Formula: C125H199N39O47S6
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Very high affinity ClC-2 blocker (apparent KD ~ 50 pM). Slows ClC-2 activation and inhibits slow-gating but does not inhibit open ClC-2 channels. Selective for ClC-2 over other ClC family members (ClC-0, ClC-1, ClC-3 and ClC-4), CFTR, GABAC, CaCC and KV1.2.
Molecular Weight: 3192, 54
