Product Overview
GR 159897 | T15415 | TargetMol Chemicals
CAS: 158848-32-9
Smiles: COC1(CS(=O)c2ccccc2)CCN(CCc2c[nH]c3ccc(F)cc23)CC1
Formula: C23H27FN2O2S
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: GR 159897 is a competitive, brain-penetrated non-peptide NK2 receptor antagonist with anti-tumor effects. GR 159897 inhibits binding of [3H]GR100679 to human NK2-CHO cells and rat colon membranes (pKis: 9.51 and 10, respectively). It can antagonize bronchoconstriction.
Molecular Weight: 414, 54
