Product Overview
GRK2-IN-1 hydrochloride (2055990-90-2 free base) | T13714L | TargetMol Chemicals
CAS: T13714L
Smiles: FC1=C(C(NCC2=NNC=C2)=O)C=C([C@H]3[C@H](COC4=CC=C(OCO5)C5=C4)CNCC3)C=C1.[H]Cl
Formula: C24H26ClFN4O4
Pathway: GPCR/G Protein
Target: GRK
Receptor: N/A
Bioactivity: GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
Molecular Weight: 488, 94
