Product Overview
GSK1016790A | T6848 | TargetMol Chemicals
CAS: 942206-85-1
Smiles: CC(C)C[C@H](NC(=O)c1cc2ccccc2s1)C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)c1ccc(Cl)cc1Cl
Formula: C28H32Cl2N4O6S2
Pathway: Membrane transporter/Ion channel|||Metabolism
Target: Calcium Channel|||TRP/TRPV Channel
Receptor: N/A
Bioactivity: GSK1016790A (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
Molecular Weight: 655, 61
