Product Overview
GSK256066 | T6054 | TargetMol Chemicals
CAS: 801312-28-7
Smiles: COc1cccc(Nc2c(cnc3c(C)cc(cc23)S(=O)(=O)c2cccc(c2)C(=O)N(C)C)C(N)=O)c1
Formula: C27H26N4O5S
Pathway: Metabolism
Target: PDE
Receptor: N/A
Bioactivity: GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380, 000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2.
Molecular Weight: 518, 59
