Product Overview
GSK256073 | T15432 | TargetMol Chemicals
CAS: 862892-90-8
Smiles: CCCCCn1c2nc(Cl)[nH]c2c(=O)[nH]c1=O
Formula: C10H13ClN4O2
Pathway: Endocrinology/Hormones|||GPCR/G Protein|||Others
Target: GPR|||Others
Receptor: N/A
Bioactivity: GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 (hydroxy-carboxylic acid receptor 2) full agonist (pEC50: 7.5). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis.
Molecular Weight: 256, 69