Product Overview
GSK343 | T6059 | TargetMol Chemicals
CAS: 1346704-33-3
Smiles: CCCc1cc(C)[nH]c(=O)c1CNC(=O)c1cc(cc2n(ncc12)C(C)C)-c1ccnc(c1)N1CCN(C)CC1
Formula: C31H39N7O2
Pathway: Autophagy|||Chromatin/Epigenetic
Target: Histone Methyltransferase|||Autophagy
Receptor: N/A
Bioactivity: GSK343, a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold specificity activity against EZH1, and >1000 fold specificity activity against other histone methyltransferases.
Molecular Weight: 541, 7
