Product Overview
GSK356278 | T27475 | TargetMol Chemicals
CAS: 720704-34-7
Smiles: CCn1ncc2c(NC3CCOCC3)c(cnc12)-c1nnc(Cc2sc(C)nc2C)o1
Formula: C21H25N7O2S
Pathway: Metabolism
Target: PDE
Receptor: N/A
Bioactivity: GSK356278 is an effective and selective inhibitor of phosphodiesterase 4 (PDE4), with pIC50s of 8.6, 8.8, and 8.7 for human PDE4A, PDE4B, and PDE4D, respectively. GSK356278 has anti-inflammatory, anxiolytic, and cognition-enhancing effects.
Molecular Weight: 439, 54