Product Overview
GSK484 hydrochloride | TQ0067 | TargetMol Chemicals
CAS: 1652591-81-5
Smiles: Cl.COC1=CC(=CC2=C1N(C)C(=N2)C1=CC2=CC=CC=C2N1CC1CC1)C(=O)N1CC[C@@H](O)[C@@H](N)C1
Formula: C27H30ClN5O3
Pathway: Chromatin/Epigenetic
Target: PAD
Receptor: N/A
Bioactivity: GSK484 hydrochloride (GTPL8577) is a specifc and reversible peptidyl arginine deiminase 4 (PAD4) inhibitor. It demonstrates high-affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium.
Molecular Weight: 510, 03