Product Overview
GYKI-52466 | T21449 | TargetMol Chemicals
CAS: 102771-26-6
Smiles: CC1=NN=C(c2ccc(N)cc2)c2cc3OCOc3cc2C1
Formula: C17H15N3O2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >50 μM for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active anticonvulsant, neuroprotective and anxiolytic in vivo.
Molecular Weight: 293, 326
